Molecular basis of specific inhibition of urokinase plasminogen activator by amiloride. [electronic resource]
Producer: 20000802Description: 109-23 p. digitalISSN:- 0305-7232
- Amiloride -- chemistry
- Amino Acid Chloromethyl Ketones -- chemistry
- Amino Acid Sequence
- Antineoplastic Agents -- chemistry
- Binding Sites -- drug effects
- Binding, Competitive
- Catalysis -- drug effects
- Crystallography, X-Ray
- Drug Design
- Humans
- Models, Molecular
- Molecular Conformation
- Molecular Sequence Data
- Neoplasm Proteins -- antagonists & inhibitors
- Protein Binding
- Protein Conformation
- Protein Structure, Tertiary
- Sequence Alignment
- Sequence Homology, Amino Acid
- Serine Proteinase Inhibitors -- chemistry
- Substrate Specificity
- Tissue Plasminogen Activator -- chemistry
- Urokinase-Type Plasminogen Activator -- antagonists & inhibitors
- Water -- chemistry
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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